Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04650
Ion Channel
Acid-sensing ion channel 3
Peptide Function
Inhibitor
Gene Name
ASIC3
Activity Data (nM)
IC50
57 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GTACSCGNSKGIYWFYRPSCPTDRGYTGSCRYFLGTCCTPAD
Peptide UniProt Accession
UniParc
UPI0000367831
Peptide Synonyms/Alias
[APETx2; 713544-47-9; H-Gly-DL-xiThr-DL-Ala-DL-Cys(1)-DL-Ser-DL-Cys(2)-Gly-DL-Asn-DL-Ser-DL-Lys-Gly-DL-xiIle-DL-Tyr-DL-Trp-DL-Phe-DL-Tyr-DL-Arg-DL-Pro-DL-Ser-DL-Cys(3)-DL-Pro-DL-xiThr-DL-Asp-DL-Arg-Gly-DL-Tyr-DL-xiThr-Gly-DL-Ser-DL-Cys(2)-DL-Arg-DL-Tyr-DL-Phe-DL-Leu-Gly-DL-xiThr-DL-Cys(1)-DL-Cys(3)-DL-xiThr-DL-Pro-DL-Ala-DL-Asp-OH; AKOS024458355]
Peptide Species
Anthopleura elegantissima (Green aggregating anemone) (Actinia elegantissima)
Peptide Name
Pi-actitoxin-Ael2b
CAS Number
713544-47-9
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−60 mV
Temperature
19–21 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
ASICs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available